4MNV | pdb_00004mnv

Crystal structure of bicyclic peptide UK729 bound as an acyl-enzyme intermediate to urokinase-type plasminogen activator (uPA)

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RCSB PDB Mol* Viewer 2.11.2 [1/27/2025, 4:56:27 PM]
Sequence of
16   ​I​​I​​G​​G​​E​​F​​T​​T​​I​​E​26   ​N​​Q​​P​​W​​F​​A​​A​​I​​Y​​R​36   ​R​​H​​R​​G​​G​​S​​V​​T​​Y​​V​42   ​C​​G​​G​​S​​L​​I​​S​​P​​C​​W​52   ​V​​I​​S​​A​​T​​H​​C​​F​​I​​D​60B  ​Y​​P​​K​​K​​E​​D​​Y​​I​​V​​Y​68   ​L​​G​​R​​S​​R​​L​​N​​S​​N​​T​78   ​Q​​G​​E​​M​​K​​F​​E​​V​​E​​N​88   ​L​​I​​L​​H​​K​​D​​Y​​S​​A​​D​97A  ​T​​L​​A​​H​​H​​N​​D​​I​​A​​L​106  ​L​​K​​I​​R​​S​​K​​E​​G​​R​​C​112  ​A​​Q​​P​​S​​R​​T​​I​​Q​​T​​I​122  ​A​​L​​P​​S​​M​​Y​​N​​D​​P​​Q​132  ​F​​G​​T​​S​​C​​E​​I​​T​​G​​F​142  ​G​​K​​E​​Q​​S​​T​​D​​Y​​L​​Y​152  ​P​​E​​Q​​L​​K​​M​​T​​V​​V​​K​162  ​L​​I​​S​​H​​R​​E​​C​​Q​​Q​​P​170B ​H​​Y​​Y​​G​​S​​E​​V​​T​​T​​K​180  ​M​​L​​C​​A​​A​​D​​P​​Q​​W​​K​188  ​T​​D​​S​​C​​Q​​G​​D​​S​​G​​G​198  ​P​​L​​V​​C​​S​​L​​Q​​G​​R​​M​208  ​T​​L​​T​​G​​I​​V​​S​​W​​G​​R​218  ​G​​C​​A​​L​​K​​D​​K​​P​​G​​V​228  ​Y​​T​​R​​V​​S​​H​​F​​L​​P​​W​238  ​I​​R​​S​​H​​T​
Type
Asm Id
Dynamic Bonds

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