Structure Determination MethodologyScientific Name of Source OrganismRefinement Resolution (Å)Enzyme Classification Name | Schaefer, M., Jautelat, R., Brumby, T., Briem, H., Eisenbrand, G., Schwahn, S., Krueger, M., Luecking, U., Prien, O., Siemeister, G. (2005) Chembiochem 6: 531 Released | 2005-03-09 | Method | X-RAY DIFFRACTION 1.9 Å | Organisms | | Macromolecule | | Unique Ligands | BRY |
Schaefer, M., Jautelat, R., Brumby, T., Briem, H., Eisenbrand, G., Schwahn, S., Krueger, M., Luecking, U., Prien, O., Siemeister, G. (2005) Chembiochem 6: 531 Released | 2005-03-09 | Method | X-RAY DIFFRACTION 2.6 Å | Organisms | | Macromolecule | | Unique Ligands | RYU |
Schaefer, M., Luecking, U., Siemeister, G., Briem, H., Krueger, M., Lienau, P., Jautelat, R. (2007) ChemMedChem 2: 63 Released | 2007-11-06 | Method | X-RAY DIFFRACTION 2.5 Å | Organisms | | Macromolecule | | Unique Ligands | PY8 |
Roehrig, S., Straub, A., Pohlmann, J., Lampe, T., Pernerstorfer, J., Schlemmer, K., Reinemer, P., Perzborn, E., Schaefer, M. (2005) J Med Chem 48: 5900-5908 Released | 2008-11-11 | Method | X-RAY DIFFRACTION 2.08 Å | Organisms | | Macromolecule | | Unique Ligands | CA, RIV |
Luecking, U., Jautelat, R., Krueger, M., Brumby, T., Lienau, P., Schaefer, M., Briem, H., Schulze, J., Hillisch, A., Reichel, A., Siemeister, G. (2013) ChemMedChem 8: 1067 Released | 2013-09-04 | Method | X-RAY DIFFRACTION 1.95 Å | Organisms | | Macromolecule | | Unique Ligands | 3I6 |
vonNussbaum, F., Li, V.M.-J., Allerheiligen, S., Anlauf, S., Baerfacker, L., Bechem, M., Delbeck, M., Fitzgerald, M.F., Gerisch, M., Gielen-Haertwig, H., Haning, H., Karthaus, D., Lang, D., Lustig, K., Meibom, D., Mittendorf, J., Rosentreter, U., Schaefer, M., Schaefer, S., Schamberger, J., Telan, L.A., Tersteegen, A. (2015) ChemMedChem 10: 1163-1173 Released | 2015-08-19 | Method | X-RAY DIFFRACTION 1.81 Å | Organisms | | Macromolecule | | Unique Ligands | JJD, NAG | Unique branched monosaccharides | FUC, NAG |
vonNussbaum, F., Li, V.M.-J., Allerheiligen, S., Anlauf, S., Baerfacker, L., Bechem, M., Delbeck, M., Fitzgerald, M.F., Gerisch, M., Gielen-Haertwig, H., Haning, H., Karthaus, D., Lang, D., Lustig, K., Meibom, D., Mittendorf, J., Rosentreter, U., Schaefer, M., Schaefer, S., Schamberger, J., Telan, L.A., Tersteegen, A. (2015) ChemMedChem 10: 1163-1173 Released | 2015-08-19 | Method | X-RAY DIFFRACTION 1.78 Å | Organisms | | Macromolecule | | Unique Ligands | EPE, JJS, NAG | Unique branched monosaccharides | FUC, NAG |
vonNussbaum, F., Li, V.M.-J., Allerheiligen, S., Anlauf, S., Baerfacker, L., Bechem, M., Delbeck, M., Fitzgerald, M.F., Gerisch, M., Gielen-Haertwig, H., Haning, H., Karthaus, D., Lang, D., Lustig, K., Meibom, D., Mittendorf, J., Rosentreter, U., Schaefer, M., Schaefer, S., Schamberger, J., Telan, L.A., Tersteegen, A. (2015) ChemMedChem 10: 1163-1173 Released | 2015-08-19 | Method | X-RAY DIFFRACTION 2.23 Å | Organisms | | Macromolecule | | Unique Ligands | DMS, JJX, NAG | Unique branched monosaccharides | FUC, NAG |
vonNussbaum, F., Li, V.M.-J., Allerheiligen, S., Anlauf, S., Baerfacker, L., Bechem, M., Delbeck, M., Fitzgerald, M.F., Gerisch, M., Gielen-Haertwig, H., Haning, H., Karthaus, D., Lang, D., Lustig, K., Meibom, D., Mittendorf, J., Rosentreter, U., Schaefer, M., Schaefer, S., Schamberger, J., Telan, L.A., Tersteegen, A. (2015) ChemMedChem 10: 1163-1173 Released | 2015-08-19 | Method | X-RAY DIFFRACTION 2.1 Å | Organisms | | Macromolecule | | Unique Ligands | JJV, MES, XPE | Unique branched monosaccharides | FUC, NAG |
vonNussbaum, F., Li, V.M., Meibom, D., Anlauf, S., Bechem, M., Delbeck, M., Gerisch, M., Harrenga, A., Karthaus, D., Lang, D., Lustig, K., Mittendorf, J., Schaefer, M., Schaefer, S., Schamberger, J. (2016) ChemMedChem 11: 199-206 Released | 2016-08-03 | Method | X-RAY DIFFRACTION 2.23 Å | Organisms | | Macromolecule | | Unique Ligands | IUY, NAG | Unique branched monosaccharides | FUC, NAG |
vonNussbaum, F., Li, V.M., Meibom, D., Anlauf, S., Bechem, M., Delbeck, M., Gerisch, M., Harrenga, A., Karthaus, D., Lang, D., Lustig, K., Mittendorf, J., Schaefer, M., Schaefer, S., Schamberger, J. (2016) ChemMedChem 11: 199 Released | 2016-08-03 | Method | X-RAY DIFFRACTION 1.9 Å | Organisms | | Macromolecule | | Unique Ligands | MES, MLI, VBM | Unique branched monosaccharides | FUC, NAG |
von Nussbaum, F., Li, V.M., Meibom, D., Anlauf, S., Bechem, M., Delbeck, M., Gerisch, M., Harrenga, A., Karthaus, D., Lang, D., Lustig, K., Mittendorf, J., Schaefer, M., Schaefer, S., Schamberger, J. (2016) ChemMedChem 11: 199-206 Released | 2016-08-03 | Method | X-RAY DIFFRACTION 2 Å | Organisms | | Macromolecule | | Unique Ligands | IUL, NAG | Unique branched monosaccharides | FUC, NAG |
von Nussbaum, F., Li, V.M., Schaefer, M. (2015) Bioorg Med Chem Lett 25: 4370-4381 Released | 2015-08-19 | Method | X-RAY DIFFRACTION 1.6 Å | Organisms | | Macromolecule | | Unique Ligands | CL, WQQ | Unique branched monosaccharides | FUC, NAG |
Schaefer, M., Scott, W.J., Hentemann, M.F., Rowley, R.B., Bull, C.O., Jenkins, S., Bullion, A.M., Johnson, J., Redman, A., Robbins, A.H., Esler, W., Fracasso, R.P., Garrison, T., Hamilton, M., Michels, M., Wood, J.E., Wilkie, D.P., Xiao, H., Levy, J., Liu, N., Stasik, E., Brands, M., Lefranc, J. (2016) ChemMedChem 11: 1517 Released | 2016-04-20 | Method | X-RAY DIFFRACTION 2.68 Å | Organisms | | Macromolecule | | Unique Ligands | 6E2, SO4 |
Schaefer, M., Buchmueller, A., Dittmer, F., Strassburger, J., Wilmen, A. (2019) J Mol Biology 431: 4817-4833 Released | 2019-09-11 | Method | X-RAY DIFFRACTION 2.7 Å | Organisms | | Macromolecule | | Unique Ligands | DMS, SO4 |
Schaefer, M., Roehrig, S., Ackerstaff, J., Nunez, E.J., Gericke, K.M., Meier, K., Tersteegen, A., Stampfuss, J., Ellerbrock, P., Meibom, D., Lang, D., Heitmeier, S., Hillisch, A. (2023) J Med Chem 66: 12203-12224 Released | 2023-09-13 | Method | X-RAY DIFFRACTION 1.841 Å | Organisms | | Macromolecule | | Unique Ligands | CIT, QV3 |
Schaefer, M., Roehrig, S., Ackerstaff, J., Nunez, E.J., Gericke, K.M., Meier, K., Tersteegen, A., Stampfuss, J., Ellerbrock, P., Meibom, M., Lang, D., Heitmeier, S., Hillisch, A. (2023) J Med Chem 66: 12203-12224 Released | 2023-09-13 | Method | X-RAY DIFFRACTION 1.75 Å | Organisms | | Macromolecule | | Unique Ligands | GOL, QVI |
Schaefer, M., Roehrig, S., Ackerstaff, J., Nunez, E.J., Gericke, K.M., Meier, K., Tersteegen, A., Stampfuss, J., Ellerbrock, P., Meibom, D., Lang, D., Heitmeier, S., Hillisch, A. (2023) J Med Chem 66: 12203-12224 Released | 2023-09-13 | Method | X-RAY DIFFRACTION 1.7 Å | Organisms | | Macromolecule | | Unique Ligands | CIT, GOL, QVO |
Schaefer, M., Roehrig, S., Ackerstaff, J., Nunez, E.J., Gericke, K.M., Meier, K., Tersteegen, A., Stampfuss, J., Ellerbrock, P., Meibom, D., Lang, D., Heitmeier, S., Hillisch, A. (2023) J Med Chem 66: 12203-12224 Released | 2023-09-13 | Method | X-RAY DIFFRACTION 1.25 Å | Organisms | | Macromolecule | | Unique Ligands | CIT, GOL, QW0 |
Schaefer, M., Roehrig, S., Ackerstaff, J., Nunez, E.J., Gericke, K.M., Meier, K., Tersteegen, A., Stampfuss, J., Ellerbrock, P., Meibom, D., Lang, D., Heitmeier, S., Hillisch, A. (2023) J Med Chem 66: 12203-12224 Released | 2023-09-13 | Method | X-RAY DIFFRACTION 1.25 Å | Organisms | | Macromolecule | | Unique Ligands | CIT, QW6, TRS |
Schaefer, M. (2024) J Med Chem 67: 17429-17453 Released | 2024-06-26 | Method | X-RAY DIFFRACTION 2 Å | Organisms | | Macromolecule | | Unique Ligands | GOL, XON |
Schaefer, M., Fuerstner, C., Ackerstaff, J., Meier, H., Straub, A., Mittendorf, J., Schamberger, J., Boerngen, K., Joerissen, H., Zubow, D., Zimmermann, K., Tersteegen, A., Geiss, V., Hartmann, E., Albrecht-Kuepper, B., Dorleans-Juste, P., Lapointe, C., Vincent, L., Heitmeier, S., Tinel, H. (2025) J Med Chem 68: 6108-6126 Released | 2024-11-27 | Method | X-RAY DIFFRACTION 2.375 Å | Organisms | | Macromolecule | | Unique Ligands | A1IJV, NAG, ZN |
Schaefer, M., Fuerstner, C. (2025) J Med Chem 68: 6108-6126 Released | 2024-11-27 | Method | X-RAY DIFFRACTION 1.987 Å | Organisms | | Macromolecule | | Unique Ligands | A1IJO, NAG, ZN | Unique branched monosaccharides | NAG |
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